Virtuelle (Nano) Welten: PDB Molecule of the Month 45: Estrogen Receptor

PDB ID	Authors	First Page	Medline Link	Journal Name	Title	Volume No	Publication Year

1A52	D.M.Tanenbaum, Y.Wang, S.P.Williams, P.B.Sigler	5998	9600906	Proc Natl Acad Sci U S A	Crystallographic comparison of the estrogen and progesterone receptor's ligand binding domains.	95	1998
1ERE	A.M.Brzozowski, A.C.Pike, Z.Dauter, R.E.Hubbard, T.Bonn, O.Engstrom, L.Ohman, G.L.Greene, J.A.Gustafsson, M.Carlquist	753	9338790	Nature	Molecular basis of agonism and antagonism in the oestrogen receptor.	389	1997
1ERR	A.M.Brzozowski, A.C.Pike, Z.Dauter, R.E.Hubbard, T.Bonn, O.Engstrom, L.Ohman, G.L.Greene, J.A.Gustafsson, M.Carlquist	753	9338790	Nature	Molecular basis of agonism and antagonism in the oestrogen receptor.	389	1997
1G50	S.Eiler, M.Gangloff, S.Duclaud, D.Moras, M.Ruff	165	( 1G50 )	Protein Expression Purif.	Overexpression, Purification, and Crystal Structure of Native Er Alpha Lbd	22	2001
1GWQ	A.Warnmark, E.Treuter, J.-A.Gustafsson, R.E.Hubbard, A.M.Brzozowski, A.C.W.Pike	21862	( 1GWQ )	J.Biol.Chem.	Interaction of Tif2 Nr-Box Peptides with the Coactivator Binding Site of Er Alpha	277	2002
1GWR	A.Warnmark, E.Treuter, J.-A.Gustafsson, R.E.Hubbard, A.M.Brzozowski, A.C.W.Pike	21862	( 1GWR )	J.Biol.Chem.	Interaction of Tif2 Nr-Box Peptides with the Coactivator Binding Site of Er Alpha	277	2002
1HCP	J.W.R.Schwabe, L.Chapman, J.T.Finch, D.Rhodes, D.Neuhaus	187	( 1HCP )	Structure	DNA RECOGNITION BY THE ESTROGEN-RECEPTOR - FROM SOLUTION TO THE CRYSTAL.	1	1993
1HCQ	J.W.Schwabe, L.Chapman, J.T.Finch, D.Rhodes	567	8221895	Cell	The crystal structure of the estrogen receptor DNA-binding domain bound to DNA: how receptors discriminate between their response elements.	75	1993
1HJ1	A.C.Pike, A.M.Brzozowski, J.Walton, R.E.Hubbard, A.G.Thorsell, Y.L.Li, J.A.Gustafsson, M.Carlquist	145	( 1HJ1 )	Structure Fold.Des.	Structural Insights Into the Mode of Action of a Pure Antiestrogen	9	2001
1KV6	H.Greschik, J.-M.Wurtz, S.Sanglier, W.Bourguet, A.Van Dorsselaer, D.Moras, J.-P.Renaud	303	( 1KV6 )	Mol. Cell	Structural and Functional Evidence for Ligand-Independent Transcriptional Activation by the Estrogen-Related Receptor 3	9	2002
1L2I	A.K.Shiau, D.Barstad, J.T.Radek, M.J.Meyers, K.W.Nettles, B.S.Katzenellenbogen, J.A.Katzenellenbogen, D.A.Agard, G.L.Greene	359	( 1L2I )	Nat.Struct.Biol.	Structural Characterization of a Subtype-Selective Ligand Reveals a Novel Mode of Estrogen Receptor Antagonism	9	2002
1L2J	A.K.Shiau, D.Barstad, J.T.Radek, M.J.Meyers, K.W.Nettles, B.S.Katzenellenbogen, J.A.Katzenellenbogen, D.A.Agard, G.L.Greene	359	( 1L2J )	Nat.Struct.Biol.	Structural Characterization of a Subtype-Selective Ligand Reveals a Novel Mode of Estrogen Receptor Antagonism	9	2002
1LO1	M.D.Gearhart, S.M.A.Holmbeck, R.M.Evans, H.J.Dyson, P.E.Wright	819	( 1LO1 )	J.Mol.Biol.	Monomeric Complex of Human Orphan Estrogen Related Receptor-2 with DNA: A Pseudo-Dimer Interface Mediates Extended Half-Site Recognition	327	2003
1NDE	B.R.Henke, T.G.Consler, N.Go, R.L.Hale, D.R.Hohman, S.A.Jones, A.T.Lu, L.B.Moore, J.T.Moore, L.A.Orband-Miller, R.G.Robinett, J.Shearin, P.K.Spearing, E.L.Stewart, P.S.Turnbull, S.L.Weaver, S.P.Williams, G.B.Wisely, M.H.Lambert	5492	( 1NDE )	J.Med.Chem.	A New Series of Estrogen Receptor Modulators that Display Selectivity for Estrogen Receptor Beta	45	2002
1QKM	A.C.W.Pike, A.M.Brzozowski, R.E.Hubbard, T.Bonn, A.-G.Thorsell, O.Engstrom, J.Ljunggren, J.-A.Gustaffson, M.Carlquist	101	( 1QKM )	Embo J.	Structure of the Ligand-Binding Domain of Oestrogen Receptor Beta in the Presence of a Partial Agonist and a Full Antagonist	18	1999
1QKN	A.C.W.Pike, A.M.Brzozowski, R.E.Hubbard, T.Bonn, A.-G.Thorsell, O.Engstrom, J.Ljunggren, J.-A.Gustaffson, M.Carlquist	101	( 1QKN )	Embo J.	Structure of the Ligand-Binding Domain of Oestrogen Receptor Beta in the Presence of a Partial Agonist and a Full Antagonist	18	1999
1QKT	M.Ruff, M.Gangloff, S.Eiler, S.Duclaud, J.M.Wurtz, M.Dino	n/a	( 1QKT )	To be Published	The Crystal Structure of an Estrogen Nuclear Receptor Mutant Suggest a Molecular Mechanism for the Agonism Antagonism Switch	n/a	n/a
1QKU	M.Ruff, M.Gangloff, S.Eiler, S.Duclaud, J.M.Wurtz, M.Dino	n/a	( 1QKU )	To be Published	The Crystal Structure of an Estrogen Nuclear Receptor Mutant Suggest a Molecular Mechanism for the Agonism Antagonism Switch	n/a	n/a
1UOM	J.Renaud, S.F.Bischoff, T.Buhl, P.Floersheim, B.Fournier, C.Halleux, J.Kallen, H.Keller, J.-M.Schlaeppi, W.Stark	2945	( 1UOM )	J.Med.Chem.	Estrogen Receptor Modulators: Identification and Structure-Activity Relationships of Potent Eralpha-Selective Tetrahydroisoquinoline Ligands	46	2003
3ERD	A.K.Shiau, D.Barstad, P.M.Loria, L.Cheng, P.J.Kushner, D.A.Agard, G.L.Greene	927	9875847	Cell	The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen.	95	1998
3ERT	A.K.Shiau, D.Barstad, P.M.Loria, L.Cheng, P.J.Kushner, D.A.Agard, G.L.Greene	927	9875847	Cell	The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen.	95	1998